Preface |
Cancer Drug Discovery and Development: New Paradigms for a New Millennium / E. A. Sausville ; J. I. Johnson ; C. M. Cragg ; S. Decker1: |
Evolutionary Biosynthesis of Anticancer Drugs / George R. Pettit2: |
Some Recent Developments in the Synthesis and SAR of Novel Taxanes / John F. Kadow ; Thomas Altstadt ; Shu-Hui Chen ; Pierre Dextraze Karen Du ; Craig Fairchild ; Jerzy Golik ; Steven Hansel ; Kathy A. Johnston ; Robert A. Kramer ; David R. Langley ; Frank Lee ; Byron Long ; Harold Mastalerz ; Carl Ouellet ; Robert Perrone ; William C. Rose ; Paul Scola ; Gene Schultz ; Andrew Staab ; Quifen May Xue ; Michael Walker ; Jen-Mei Wei ; Mark Wittman ; J. J. Kim Wright ; Mary Zoeckler ; Dolatrai M. Yvas3: |
New Generation Taxoids and Hybrids of Microtube-Stabilizing Anticancer Agents / Iwao Ojima ; Scott D. Kuduk ; Subrata Chakravarty ; Songnian Lin ; Tao Wang ; Xudong Geng ; Michael L. Miller ; Pierre-Yves Bounaud ; Young Hoon Park ; Cuhung-Ming Sun ; John C. Slater ; Tadashi Inoue ; Christopher P. Borella ; John J. Walsh ; Ralph J. Bernacki ; Paula Pera ; Jean Veith ; Ezio Bombzrdelli ; Antonella Riva ; Srinivasa Rao ; Hifeng He ; George A. Orr ; Susan B. Horwitz ; Samuel J. Danishefsky ; Giovanni Scambia ; Cristiano Ferlini4: |
Discodermolide and Taxol: A Synergistic Drug Combination in Human Carcinoma Cell Lines / Susan Band Horwitz ; Laura A. Martello ; Chia-Ping Y. Yang ; Amos B. Smith ; III ; Hayley M. McDaid5: |
Highly Efficient Semisynthesis of Biologically Active Epothilone Derivatives / Gregory D. Vite ; Robert M. Borzilleri ; Soong-Hoon Kim ; Alicia Regueiro-Ren ; W. Griffith Humphreys ; Francis Y. F. Lee6: |
Synthetic and Semisynthetic Analogs of Epothilones: Chemistry and Biological Activity / Karl-Heinz Altmann ; Marcel J. J. Blommers ; Giorgio Caravatti ; Andreas Florsheimer ; Kyriacos C. Nicolaou ; Terrence O'Reilly ; Alfred Schmidt ; Dieter Schinzer ; Markus Wartmann7: |
Synthesis and Biological Activity of Epothilones / Ulrich Klar ; Werner Skuballa ; Bernd Buchmann ; Wolfgang Schwede ; Thomas Bunte ; Jens Hoffmann ; Rosemarie B. Lichtner8: |
Epothelones and Sarcodictyins: From Combinatorial to Designed Analogs / Nicolas Winssinger and K. C. Nicolaou9: |
Synthesis and Structure-Activity Relationship Studies of Cryptophycins: A Novel Class of Potent Antimitotic Tumor Depsipeptides / Chuan Shih ; Rima S. Al-Awar ; Andrew H. Fray ; Michael J. Martinelli ; Eric D. Moher ; Bryan H. Norman ; Vinod F. Patel ; Richard M. Schultz ; John E. Toth ; David L. Varie ; Thomas H. Corbett ; Richard E. Moore10: |
Farnesyltransferase Inhibitors as Potential Anticancer Agents / J. B. Gibbs ; N. J. Anthony ; I. Bell ; C. A. Buser ; J. P. Davide ; S. J. deSolms ; C. Dinsmore ; S. L. Graham ; G. D. Hartman ; D. C. Heimbrook ; H. Huber ; K. S. Koblan ; N. E. Kohl ; R. B. Lobell ; T. M. Williams11: |
Farnesyltransferase Inhibitors: From Squalene Synthase Inhibitors to the Clinical Agent BMS-214662 / John T. Hunt12: |
Inhibiting Farnesyl Protein Transferase with Sch-66336: Potentially a Selective Non-Cytotoxic herapy for Human Cancer / A. G. Taveras ; F. G. Njoroge ; R. J. Doll ; J. Kelly ; S. Remiszewski ; A. K. Mallams ; C. S. Alvarez ; J. del Rosario ; R. R. Rossman ; B. Vibulbhan ; P. Pinto ; J. Deskus ; M. Connolly ; J. Wang ; J. Desai ; R. Wolin ; A. Afonso ; A. B. Cooper ; D. F. Rane ; Y.-T. Liu ; C. J. Aki ; J. Chao ; C. Strickland ; P. Weber ; M. Liu ; M. S. Bryant ; A. A. Nomeir ; R. Patton ; L. Wang ; L. James ; D. Carr ; P. Kirschmeier ; W. R. Bishop ; V. Girijavallabhan ; A. K. Ganguly13: |
Pyrrolo[2,3-d]pyrimidine and Pyrazolo[3,4-d]pyrimidine Derivatives as Selective Inhibitors of the EGF Receptor Tyrosine Kinase / G. Caravatti ; J. Bruggen ; E. Buchdunger ; R. Cozens ; P. Furet ; N. Lydon ; T. O'Reilly ; P. Traxler14: |
STI571: A New Treatment Modality for CML / Jurg Zimmermann ; Pascal Furet ; Elisabeth Buchdunger15: |
The Discovery and De / 16: |
Preface |
Cancer Drug Discovery and Development: New Paradigms for a New Millennium / E. A. Sausville ; J. I. Johnson ; C. M. Cragg ; S. Decker1: |
Evolutionary Biosynthesis of Anticancer Drugs / George R. Pettit2: |
Some Recent Developments in the Synthesis and SAR of Novel Taxanes / John F. Kadow ; Thomas Altstadt ; Shu-Hui Chen ; Pierre Dextraze Karen Du ; Craig Fairchild ; Jerzy Golik ; Steven Hansel ; Kathy A. Johnston ; Robert A. Kramer ; David R. Langley ; Frank Lee ; Byron Long ; Harold Mastalerz ; Carl Ouellet ; Robert Perrone ; William C. Rose ; Paul Scola ; Gene Schultz ; Andrew Staab ; Quifen May Xue ; Michael Walker ; Jen-Mei Wei ; Mark Wittman ; J. J. Kim Wright ; Mary Zoeckler ; Dolatrai M. Yvas3: |
New Generation Taxoids and Hybrids of Microtube-Stabilizing Anticancer Agents / Iwao Ojima ; Scott D. Kuduk ; Subrata Chakravarty ; Songnian Lin ; Tao Wang ; Xudong Geng ; Michael L. Miller ; Pierre-Yves Bounaud ; Young Hoon Park ; Cuhung-Ming Sun ; John C. Slater ; Tadashi Inoue ; Christopher P. Borella ; John J. Walsh ; Ralph J. Bernacki ; Paula Pera ; Jean Veith ; Ezio Bombzrdelli ; Antonella Riva ; Srinivasa Rao ; Hifeng He ; George A. Orr ; Susan B. Horwitz ; Samuel J. Danishefsky ; Giovanni Scambia ; Cristiano Ferlini4: |
Discodermolide and Taxol: A Synergistic Drug Combination in Human Carcinoma Cell Lines / Susan Band Horwitz ; Laura A. Martello ; Chia-Ping Y. Yang ; Amos B. Smith ; III ; Hayley M. McDaid5: |